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I. et al., \"Studies With Deuterated Drugs,\" Journal of Pharmaceutical Sciences, 1975, vol. 64 (3), pp. 367-391.","npl_type":"a","external_id":["10.1002/jps.2600640306","1151621"],"record_lens_id":"049-214-828-980-62X","lens_id":["117-512-385-237-676","049-214-828-980-62X","162-641-723-845-483"],"sequence":77,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":5,"text":"Brickner, S.J. et al., \"Synthesis And Antibacterial Activity Of U-100592 And U-100766, Two Oxazolidinone Antibacterial Agents for the Potential Treatment of Multidrug- Resistant Gram-Positive Bacterial Infections,\" Journal of Medicinal Chemistry, 1996, vol. 39 (3), pp. 673-679.","npl_type":"a","external_id":["10.1021/jm9509556","8576909"],"record_lens_id":"075-842-203-736-897","lens_id":["089-834-132-022-763","075-842-203-736-897","086-663-999-689-162"],"sequence":78,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":6,"text":"Bruncko M., et al., \"Studies Leading to Potent, Dual Inhibitors of Bcl-2 And Bcl-XL,\" Journal of Medicinal Chemistry, 2007, vol. 50 (4), pp. 641-662.","npl_type":"a","external_id":["17256834","10.1021/jm061152t"],"record_lens_id":"022-947-416-700-263","lens_id":["032-957-797-661-094","022-947-416-700-263","105-030-296-979-486"],"sequence":79,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":7,"text":"Certo M., et al., \"Mitochondria Primed by Death Signals Determine Cellular Addiction to Antiapoptotic Bcl-2 Family Members,\" Cancer Cell, 2006, vol. 9 (5), pp. 351-365.","npl_type":"a","external_id":["10.1016/j.ccr.2006.03.027","16697956"],"record_lens_id":"027-049-145-189-682","lens_id":["187-374-454-859-230","027-049-145-189-682","037-127-658-338-974"],"sequence":80,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":8,"text":"Cross, L.C. et al., \"IUPAC Commission on Nomenclature of Organic Chemistry: Rules for the Nomenclature of Organic Chemistry, Section E: Stereochemistry,\" Pure and Applied Chemistry, 1976, vol. 45, pp. 11-30.","npl_type":"a","external_id":["10.1351/pac197645010011"],"record_lens_id":"180-631-728-571-083","lens_id":["180-631-728-571-083","039-510-760-860-958"],"sequence":81,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":9,"text":"Czajka, D. M. et al., \"Effect of Deuterium Oxide on the Reproductive Potential of Mice,\" Annals of the New York Academy of Sciences, 1960, vol. 84, pp. 770-779.","npl_type":"a","external_id":["13719049","10.1111/j.1749-6632.1960.tb39109.x"],"record_lens_id":"007-913-191-371-892","lens_id":["105-675-795-798-338","007-913-191-371-892","131-119-635-533-010"],"sequence":82,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":10,"text":"Czajka, D. M. et al., \"Physiological Effects of Deuterium on Dogs,\" American Journal of Physiology, 1961, vol. 201 (2), pp. 357-362.","npl_type":"a","external_id":["10.1152/ajplegacy.1961.201.2.357","13719048"],"record_lens_id":"014-213-884-274-004","lens_id":["031-219-492-596-526","014-213-884-274-004","135-094-533-638-863"],"sequence":83,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":11,"text":"Del Gaizo Moore V., et al., \"BCL-2 Dependence and ABT-737 Sensitivity in Acute Lymphoblastic Leukemia,\" Blood, 2008, vol. 111 (4), pp. 2300-2309.","npl_type":"a","external_id":["10.1182/blood-2007-06-098012","18056841","pmc2234061"],"record_lens_id":"024-437-144-140-823","lens_id":["112-919-904-640-866","183-040-288-358-397","024-437-144-140-823"],"sequence":84,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":12,"text":"Eliel, E. L. et al., \"Stereochemistry of Organic Compounds,\" 1994, pp. 119-120, 1206, John Wiley & Sons, Inc. New York. Table of Contents.","npl_type":"a","external_id":[],"lens_id":[],"sequence":85,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":13,"text":"Foster, A. B. et al., \"Deuterium Isotope Effects in the Metabolism of Drugs and Xenobiotics: Implications for Drug Design,\" Advances in Drug Research, 1985, vol. 14, pp. 2-36.","npl_type":"a","external_id":[],"lens_id":[],"sequence":86,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":14,"text":"Harada H., et al., \"Survival Factor-Induced Extracellular Signal-Regulated Kinase Phosphorylates Bim, Inhibiting Its Association with Bax and Proapoptotic Activity,\" Proceedings of the National Academy of Sciences, 2004, vol. 101 (43), pp. 15313-15317.","npl_type":"a","external_id":["10.1073/pnas.0406837101","pmc524459","15486085"],"record_lens_id":"062-402-667-173-77X","lens_id":["197-904-692-733-033","062-402-667-173-77X","199-489-621-976-422"],"sequence":87,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":15,"text":"Holzelova, E. et al., \"Autoimmune Lymphoproliferative Syndrome with Somatic Fas Mutations,\" New England Journal of Medicine, 2004, vol. 351 (14), pp. 1409-1418.","npl_type":"a","external_id":["15459302","10.1056/nejmoa040036"],"record_lens_id":"029-731-136-159-478","lens_id":["035-170-871-997-873","029-731-136-159-478","105-675-042-354-193"],"sequence":88,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":16,"text":"International Search Report for Application No. For PCT/US2010/036919, mailed Aug. 19, 2010, 5 pages.","npl_type":"a","external_id":[],"lens_id":[],"sequence":89,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":17,"text":"International Search Report for Application No. PCT/US2009/066722, Mailed on Aug.4, 2010, 4 pages.","npl_type":"a","external_id":[],"lens_id":[],"sequence":90,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":18,"text":"International Search Report for Application No. PCT/US2009/066790, mailed on Jul. 28, 2010, 5 pages.","npl_type":"a","external_id":[],"lens_id":[],"sequence":91,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":19,"text":"International Search Report for Application No. PCT/US2010/036844, mailed on Aug. 16, 2010, 5 pages.","npl_type":"a","external_id":[],"lens_id":[],"sequence":92,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":20,"text":"Jones, C.D. et al., \"Effects of Substituent Modification on Face Selection in Reduction,\" Journal of Organic Chemistry, 1998, vol. 63 (8), pp. 2758-2760.","npl_type":"a","external_id":["11672152","10.1021/jo9721296"],"record_lens_id":"069-363-262-996-810","lens_id":["155-259-942-819-823","069-363-262-996-810","087-312-048-476-788"],"sequence":93,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":21,"text":"Kato, S. et al., \"Synthesis of Deuterated Mosapride Citrate,\" Journal of Labelled Compounds and Radiopharmaceuticals, 1995, vol. 36 (10), pp. 927-932.","npl_type":"a","external_id":["10.1002/jlcr.2580361004"],"record_lens_id":"063-434-787-171-827","lens_id":["159-594-177-361-555","063-434-787-171-827"],"sequence":94,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":22,"text":"Korolkovas A., \"Development of Drugs\" in: Essentials of Medicinal Chemistry, Second Edition, John Wiley and Sons, 1988, pp. 97-118.","npl_type":"a","external_id":[],"lens_id":[],"sequence":95,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":23,"text":"Kushner et al., \"Pharmacological uses and perspectives of heavy water and deuterated compounds,\" Canadian Journal of Physiology and Pharmacology, 1999, vol. 77 (2), pp. 79-88.","npl_type":"a","external_id":["10535697","10.1139/y99-005","10.1139/cjpp-77-2-79"],"record_lens_id":"040-081-313-970-111","lens_id":["113-879-841-341-959","040-081-313-970-111","185-003-261-063-628","151-747-747-821-255","100-689-891-218-634"],"sequence":96,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":24,"text":"Lizondo, J. et al., \"Linezolid: Oxazolidinone antibacterial,\" Drugs of the Future, 1996, vol. 21 (11), pp. 1116-1123.","npl_type":"a","external_id":["10.1358/dof.1996.021.11.383118"],"record_lens_id":"053-125-588-187-197","lens_id":["053-125-588-187-197","111-468-274-861-130"],"sequence":97,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":25,"text":"Mallesham, B. et al., \"Highly Efficient Cui-Catalyzed Coupling of Aryl Bromides With Oxazolidinones Using Buchwald's Protocol: A Short Route to Linezolid and Toloxatone,\" Organic Letters, 2003, vol. 5 (7), pp. 963-965.","npl_type":"a","external_id":["12659549","10.1021/ol026902h"],"record_lens_id":"006-794-777-498-57X","lens_id":["119-250-085-691-960","006-794-777-498-57X","103-495-342-054-351"],"sequence":98,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":26,"text":"Mason K.D., et al, \"Programmed anuclear cell death delimits platelet life span,\" Cell, 2007, vol. 128 (6), pp. 1173-1186.","npl_type":"a","external_id":["17382885","10.1016/j.cell.2007.01.037"],"record_lens_id":"008-882-258-810-261","lens_id":["078-528-859-458-002","008-882-258-810-261","113-318-470-839-239"],"sequence":99,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":27,"text":"Park C.M., et al. \"Discovery of an Orally Bioavailable Small Molecule Inhibitor of Prosurvival B-Cell Lymphoma 2 Proteins,\" Journal of Medicinal Chemistry, 2008, vol. 51 (21), pp. 6902-6915.","npl_type":"a","external_id":["10.1021/jm800669s","18841882"],"record_lens_id":"045-085-212-564-755","lens_id":["109-544-602-777-289","175-153-725-439-63X","045-085-212-564-755"],"sequence":100,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":28,"text":"Puck J.M., et al., \"Immune Disorders Caused by Defects in the Caspase Cascade ,\" Current Allergy and Asthma Reports, 2003, vol. 3, pp. 378-384.","npl_type":"a","external_id":["10.1007/s11882-003-0070-1","12906772"],"record_lens_id":"033-314-697-198-853","lens_id":["067-676-190-011-289","033-314-697-198-853","097-072-275-932-248"],"sequence":101,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":29,"text":"Rengan R., et al., \"Actin Cytoskeletal Function is Spared, but Apoptosis is Increased, in Was Patient Hematopoietic Cells,\" Blood, 2000, vol. 95 (4), pp. 1283-1292.","npl_type":"a","external_id":["10666201","10.1182/blood.v95.4.1283.004k44_1283_1292"],"record_lens_id":"006-042-988-227-006","lens_id":["089-983-668-292-568","006-042-988-227-006","069-016-410-349-177"],"sequence":102,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":30,"text":"Shimazaki K., et al., \"Evaluation of Apoptosis as a Prognostic Factor in Myelodysplastic Syndromes,\" British J Haematology, 2000, vol. 110 (3), pp. 584-590.","npl_type":"a","external_id":["10.1046/j.1365-2141.2000.02228.x","10997968"],"record_lens_id":"089-316-616-931-920","lens_id":["128-645-220-872-549","089-316-616-931-920","132-867-456-272-345"],"sequence":103,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":31,"text":"Sutton, V.R. et al., \"Bcl-2 Prevents Apoptosis Induced By Perforin And Granzyme B, But Not That Mediated By Whole Cytotoxic Lymphocytes,\" Journal of Immunology, 1997, vol. 158 (12), pp. 5783-5790.","npl_type":"a","external_id":["9190929","10.4049/jimmunol.158.12.5783"],"record_lens_id":"007-856-972-371-459","lens_id":["178-213-114-754-463","007-856-972-371-459","046-847-503-157-505"],"sequence":104,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":32,"text":"Thomson, J.F., \"Physiological Effects Of D20 in Mammals,\" Annals of the New York Academy of Sciences, 1960, vol. 84, pp. 736-744.","npl_type":"a","external_id":["10.1111/j.1749-6632.1960.tb39105.x","13776654"],"record_lens_id":"068-656-513-877-430","lens_id":["089-488-158-658-007","068-656-513-877-430","150-120-950-715-794"],"sequence":105,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":33,"text":"Tse, C. et al., \"ABT-263: A Potent and Orally Bioavailable Bcl-2 Family Inhibitor,\" Cancer Research, 2008, vol. 68 (9), pp. 3421-3428-Including Supplementary Data.","npl_type":"a","external_id":["10.1158/0008-5472.can-07-5836","18451170"],"record_lens_id":"016-735-453-562-734","lens_id":["048-950-137-852-177","045-928-373-581-970","016-735-453-562-734"],"sequence":106,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":34,"text":"Wang, Z. X., \"An Exact Mathematical Expression for Describing Competitive Binding of Two Different Ligands to a Protein Molecule,\" FEBS Letters, 1995, vol. 360 (2), pp. 111- 114.","npl_type":"a","external_id":["10.1016/0014-5793(95)00062-e","7875313"],"record_lens_id":"074-633-529-904-195","lens_id":["170-243-533-082-610","074-633-529-904-195","172-611-454-633-866"],"sequence":107,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":35,"text":"Wendt M., \"Discovery of ABT-263, a Bcl-Family Protein Inhibitor: Observations on Targeting a Large Protein-Protein Interaction,\" Expert Opinion on Drug Discovery , 2008, vol. 3 (9), pp. 1123-1143.","npl_type":"a","external_id":["23506184","10.1517/17460441.3.9.1123"],"record_lens_id":"114-558-137-490-394","lens_id":["175-232-523-008-036","171-251-818-372-765","114-558-137-490-394"],"sequence":108,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":36,"text":"Written Opinion for Application No. PCT/US2007/077579, mailed on Jul.29, 2008, 9 pages.","npl_type":"a","external_id":[],"lens_id":[],"sequence":109,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":37,"text":"Written Opinion of the International Searching Authority for Application No. PCT/US2010/036844, 10 pages.","npl_type":"a","external_id":[],"lens_id":[],"sequence":110,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":38,"text":"Written Opinion of the International Searching Authority for Application No. PCT/US2010/036919, 9 pages.","npl_type":"a","external_id":[],"lens_id":[],"sequence":111,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":39,"text":"Zhang H., et al., \"Bc1-2 Family Proteins are Essential for Platelets Survival,\" Cell Death and Differentiation, 2007, vol. 14 (5), pp. 943-951.","npl_type":"a","external_id":["17205078","10.1038/sj.cdd.4402081"],"record_lens_id":"000-677-079-761-288","lens_id":["025-462-919-814-426","000-677-079-761-288","197-513-929-056-328"],"sequence":112,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":40,"text":"Sophie A., et al., \"Synthesis of \"Trioxaquantel\" Derivatives as Potential New Antischistosomal Drugs,\" European Journal of Organic Chemistry, 2008, vol. 5, pp. 895-913.","npl_type":"a","external_id":[],"lens_id":[],"sequence":113,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":41,"text":"International Search Report for Application No. PCT/US2010/057587, mailed on Apr. 28, 2011, 4 pages.","npl_type":"a","external_id":[],"lens_id":[],"sequence":114,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":42,"text":"ISA, International Search Report dated Feb. 9, 2011 for PCT/US2010/036198.","npl_type":"a","external_id":[],"lens_id":[],"sequence":115,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":43,"text":"ISA, PCT Written Opinion of the International Search Authority dated Feb. 9, 2011 for PCT/US2010/036198.","npl_type":"a","external_id":[],"lens_id":[],"sequence":116,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":44,"text":"ISA, Supplementary International Search Report dated Sep. 8, 2011 for PCT/US2010/036198.","npl_type":"a","external_id":[],"lens_id":[],"sequence":117,"category":[],"us_category":[],"cited_phase":"APP","rel_claims":[]}},{"npl":{"num":45,"text":"Skoug et al. Enabling Discovery Through Formulation. American Association of Pharmaceutical Scientists (AAPS) Webinar [online]). Presented Mar. 18, 2010, 12:30 PM to 2:00 PM EDT. Obtained from webinar conductors. For information see
methyl trans-4-{[(4-{[4-(4-{[2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoyl]sulfamoyl}-2-nitrophenyl)amino]methyl}cyclohexanecarboxylate;\n
trans-4-{[(4-{[4-(4-{[2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoyl]sulfamoyl}-2-nitrophenyl)amino]methyl}cyclohexanecarboxylic acid;\n
N-(4-{[4-(4-{[2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoyl]sulfamoyl}-2-nitrophenyl)-4-cyanopiperidine-1-carboxamide;\n
4-(4-{[2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-N-{[4-({[cis-4-(methoxymethyl)cyclohexyl]methyl}amino)-3-nitrophenyl]sulfonyl}-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide;\n
4-(4-{[2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-N-{[4-({[trans-4-(methoxymethyl)cyclohexyl]methyl}amino)-3-nitrophenyl]sulfonyl}-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide;\n
4-(4-{[2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)-N-{[1-(tetrahydro-2H-pyran-4-ylmethyl)-1H-benzotriazol-5-yl]sulfonyl}benzamide;\n
N-({5-chloro-6-[(2-oxo-1-oxa-3-azaspiro[4.5]dec-8-yl)methoxy]pyridin-3-yl}sulfonyl)-4-(4-{[2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide;\n
N-(4-{[4-(4-{[2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoyl]sulfamoyl}-2-nitrophenyl)-4-methoxypiperidine-1-carboxamide;\n
N-({5-chloro-6-[(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-5-yl)methoxy]pyridin-3-yl}sulfonyl)-4-(4-{[2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide;\n
4-(4-{[2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)-N-{[1-(tetrahydro-2H-pyran-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-5-yl]sulfonyl}benzamide;\n
4-(4-{[2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-N-{[3-chloro-1-(tetrahydro-2H-pyran-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-5-yl]sulfonyl}-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide\n
4-(4-{[2-(4-chlorophenyl)-4-(methoxymethyl)-4-methylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-N-({3-nitro-4-[(tetrahydro-2H-pyran-4-ylmethyl)amino]phenyl}sulfonyl)-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide;\n
N-[(4-{[4,4-bis(hydroxymethyl)cyclohexyl]methoxy}-3-nitrophenyl)sulfonyl]-4-(4-{[2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide;\n
N-(2-chloro-4-{[4-(4-{[2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoyl]sulfamoyl}phenyl)-4-methoxypiperidine-1-carboxamide;\n
N-(2-chloro-4-{[4-(4-{[2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoyl]sulfamoyl}phenyl)-4-cyanopiperidine-1-carboxamide;\n
N-(2-chloro-4-{[4-(4-{[2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoyl]sulfamoyl}phenyl)-4-hydroxy-4-methylpiperidine-1-carboxamide;\n
N-(2-chloro-4-{[4-(4-{[2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoyl]sulfamoyl}phenyl)-4-(methoxymethyl)piperidine-1-carboxamide;\n
N-[(5-chloro-6-{[(5r,8r)-2-oxo-1-oxa-3-azaspiro[4.5]dec-8-yl]methoxy}pyridin-3-yl)sulfonyl]-4-(4-{[2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide;\n
N-[(5-chloro-6-{[(5s,8s)-2-oxo-1-oxa-3-azaspiro[4.5]dec-8-yl]methoxy}pyridin-3-yl)sulfonyl]-4-(4-{[2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide;\n
N-(2-chloro-4-{[4-(4-{[2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoyl]sulfamoyl}phenyl)-4-(morpholin-4-yl)piperidine-1-carboxamide;\n
N-[(5-chloro-6-{[trans-4-hydroxy-4-(methoxymethyl)cyclohexyl]methoxy}pyridin-3-yl)sulfonyl]-4-(4-{[2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide;\n
N-[(5-chloro-6-{[cis-4-hydroxy-4-(hydroxymethyl)cyclohexyl]methoxy}pyridin-3-yl)sulfonyl]-4-(4-{[2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide;\n
N-[(5-chloro-6-{[trans-4-hydroxy-4-(hydroxymethyl)cyclohexyl]methoxy}pyridin-3-yl)sulfonyl]-4-(4-{[2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide;\n
N-[(5-chloro-6-{[4-fluoro-1-(oxetan-3-yl)piperidin-4-yl]methoxy}pyridin-3-yl)sulfonyl]-4-(4-{[2-(4-chlorophenyl)-5-methoxy-5-methylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide;\n
4-(4-{[2-(4-chlorophenyl)cyclohex-1-en-1-yl]methyl}piperazin-1-yl)-N-({3-nitro-4-[(tetrahydro-2H-pyran-4-ylmethyl)amino]phenyl}sulfonyl)-2-(1H-pyrrolo pyridin-5-yloxy)benzamide;\n
4-(4-chlorophenyl)-1-methyl-3-[(4-{4-[({3-nitro-4-[(tetrahydro-2H-pyran-4-ylmethyl)amino]phenyl}sulfonyl)carbamoyl]-3-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)phenyl}piperazin-1-yl)methyl]cyclohex-3-ene-1-carboxylic acid; and\n
N-[(5-chloro-6-{[1-(oxetan-3-yl)piperidin-4-yl]methoxy}pyridin-3-yl)sulfonyl]-4-(4-{[2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide."],"number":1,"annotation":false,"claim":true,"title":false},{"lines":["N-[(5-chloro-6-{[trans-4-hydroxy-4-(methoxymethyl)cyclohexyl]methoxy}pyridin-3-yl)sulfonyl]-4-(4-{[2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide, or a pharmaceutically acceptable salt thereof."],"number":2,"annotation":false,"claim":true,"title":false},{"lines":["A composition for treating lymphoblastic leukemia, said composition comprising an excipient and a therapeutically effective amount of the compound or pharmaceutically acceptable salt of claim 1 or claim 2."],"number":3,"annotation":false,"claim":true,"title":false}]}},"filters":{"npl":[],"notNpl":[],"applicant":[],"notApplicant":[],"inventor":[],"notInventor":[],"owner":[],"notOwner":[],"tags":[],"dates":[],"types":[],"notTypes":[],"j":[],"notJ":[],"fj":[],"notFj":[],"classIpcr":[],"notClassIpcr":[],"classNat":[],"notClassNat":[],"classCpc":[],"notClassCpc":[],"so":[],"notSo":[],"sat":[]},"sequenceFilters":{"s":"SEQIDNO","d":"ASCENDING","p":0,"n":10,"sp":[],"si":[],"len":[],"t":[],"loc":[]}}