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PROBLEM TO BE SOLVED: To provide a new immunosuppressor which has pharmacological activity similar to that of the natural compound cyclosporine A without exhibiting adverse effects.
SOLUTION: The above problem is solved by providing pharmacologically effective several mixtures of cis- and trans-isomers of cyclosporine A analogues. This invention relates to an isomer mixture of cyclosporine analogues structurally-similar to cyclosporine A. These mixtures exhibit a higher effect and lower toxicity in comparison with each isomer and with natural and other cyclosporines and cyclosporine derivatives, both heretofore known currently. The examples of this invention relates to cyclosporine A analogues called ISA
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